SCHEMBL8403207

SCHEMBL8403207

Cc1ccc2c(c1)/C(=N/O)CCC2C1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
RAB9A P51151 6/20 0.36
NPC1 O15118 5/20 0.36
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
KMT2A Q03164 3/20 0.36
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
MEN1 O00255 2/20 0.32
SRD5A1 P18405 2/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
LMNA P02545 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8403210 1.00 ALDH1A1 (0.39) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL8400995 0.80 ALDH1A1 (0.51) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL8920864 0.80 HPGD (0.44) MAPTSMN1; SMN2KMT2ANPSR1MEN1
SCHEMBL8920861 0.80 HPGD (0.44) MAPTSMN1; SMN2KMT2ANPSR1MEN1
SCHEMBL8402982 0.77 NPC1 (0.35) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL8402981 0.77 NPC1 (0.35) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL8402475 0.77 KDM4E (0.31) RAB9ANPC1SMN1; SMN2KMT2ATSHR
SCHEMBL8402477 0.77 KDM4E (0.31) RAB9ANPC1SMN1; SMN2KMT2ATSHR
SCHEMBL8398673 0.74 SLC6A2 (0.38) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL8399422 0.72 SLC6A2 (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711283-B1 TETRAHYDRO-1H-BENZAZEPINONES AND HEXAHYDROAZEPINONES AS SELECTIVE CHOLECYSTOKININ-B RECEPTOR ANTAGONISTS PFIZER (US) 1999-06-16 EP disclosed
US-5618811-A Tetrahydro-1H-benzazepinones and hexahydroazepinones as selective cholecystokinin-B receptor antagonists PFIZER INC. (US) 1997-04-08 US disclosed