SCHEMBL8405359

SCHEMBL8405359

Oc1cc(Cl)c(OCCCOc2ccc(C(F)(F)F)cc2)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.43
PPARD Q03181 2/20 0.43
RHOC P08134 1/20 0.42
RHOA P61586 1/20 0.42
MAOB P27338 5/20 0.41
NOS1 P29475 2/20 0.41
PTGS1 P23219 1/20 0.41
THRB P10828 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.40
LTA4H P09960 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8405863 0.97 NOS1 (0.43) PPARAPPARDRHOCRHOAMAOB
SCHEMBL8408847 0.91 PPARA (0.42) PPARAPPARDRHOCRHOAMAOB
SCHEMBL8409110 0.88 PPARA (0.45) PPARAPPARDRHOCRHOA
SCHEMBL8406354 0.88 PPARA (0.40) PPARAPPARDRHOCRHOAMAOB
SCHEMBL8405443 0.85 PPARA (0.42) PPARAPPARDRHOCRHOALTA4H
SCHEMBL8405614 0.85 FFAR4 (0.47) PPARAPPARDMAOBMRGPRX4
SCHEMBL8407208 0.85 HRH3 (0.43)
SCHEMBL8409230 0.84 MAOB (0.40) PPARDMAOBPTGS1THRBMRGPRX4
SCHEMBL8408886 0.84 FFAR4 (0.38) PPARAPPARDRHOCRHOALTA4H
SCHEMBL8405716 0.83 POLB (0.48) PPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP claimed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP claimed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO claimed
US-5872137-A AROMATIC OXY DIHALOPRENE COMPOUNDS INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-02-16 US disclosed
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP disclosed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP disclosed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO disclosed