SCHEMBL8407972

SCHEMBL8407972

COC(=O)NC(=N)c1ccc(-c2ccc(C(=O)NC3CCC(C(=O)OC)CC3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.51
RAB9A P51151 4/20 0.51
NPC1 O15118 3/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
SMYD3 Q9H7B4 3/20 0.46
HPGD P15428 2/20 0.41
MAPK14 Q16539 5/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
FYN P06241 1/20 0.41
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN11 Q06124 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP2C9 P11712 2/20 0.40
CFTR P13569 1/20 0.40
MAPT P10636 1/20 0.39
CYP46A1 Q9Y6A2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9568208 0.85 SCN1A (0.44) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL9568210 0.85 SCN1A (0.44) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL9185970 0.85 MEN1 (0.54) SMN1; SMN2RAB9ANPC1MEN1KMT2A
Hydrochloric Acid SCHEMBL8410586 0.84 MEN1 (0.52) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL8949258 0.79 CNR2 (0.41) SMN1; SMN2RAB9AMEN1KMT2AHPGD
SCHEMBL8949056 0.79 CNR2 (0.41) SMN1; SMN2RAB9AMEN1KMT2AHPGD
SCHEMBL8409339 0.79 NPC1 (0.61) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL9174248 0.78 MAPT (0.48) SMN1; SMN2MEN1KMT2ASMYD3HPGD
SCHEMBL15498625 0.77 MEN1 (0.59) SMN1; SMN2RAB9ANPC1MEN1KMT2A
SCHEMBL15510848 0.77 MEN1 (0.59) SMN1; SMN2RAB9ANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed