SCHEMBL8409016

SCHEMBL8409016

Oc1cc(Cl)c(OCc2cccc(Oc3cc(Cl)cc(Cl)c3)c2)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.47
FFAR1 O14842 3/20 0.40
FFAR4 Q5NUL3 1/20 0.40
FAAH O00519 1/20 0.40
NR4A2 P43354 1/20 0.40
FDFT1 P37268 1/20 0.40
HSP90AA1 P07900 1/20 0.40
MAOB P27338 3/20 0.39
MAOA P21397 1/20 0.39
RXRA P19793 2/20 0.38
RXRB P28702 2/20 0.38
RXRG P48443 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8405973 0.89 PPARG (0.47) MRGPRX4FFAR1FFAR4NR4A2MAOB
SCHEMBL8405485 0.89 FFAR1 (0.51) MRGPRX4FFAR1FFAR4
SCHEMBL8409040 0.86 HSP90AA1 (0.54) MRGPRX4FFAR1FFAR4FAAHFDFT1
SCHEMBL8408975 0.84 FFAR1 (0.55) MRGPRX4FFAR1FFAR4MAOB
SCHEMBL8408818 0.84 FFAR1 (0.44) MRGPRX4FFAR1FFAR4FAAHNR4A2
SCHEMBL8405460 0.83 MRGPRX4 (0.43) MRGPRX4FFAR1FFAR4FAAHNR4A2
SCHEMBL8408376 0.81 CYP4F2 (0.56) MRGPRX4FFAR1NR4A2MAOBMAOA
SCHEMBL8405447 0.81 MAOB (0.54) MRGPRX4MAOB
SCHEMBL8405474 0.81 NR4A1 (0.43) FFAR1FFAR4FAAHNR4A2FDFT1
SCHEMBL8407398 0.81 CYP3A4 (0.53) MRGPRX4NR4A2HSP90AA1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5872137-A AROMATIC OXY DIHALOPRENE COMPOUNDS INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-02-16 US disclosed
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP disclosed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP disclosed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO disclosed