SCHEMBL8409033

SCHEMBL8409033

CCOC(=O)CCNC(=O)Nc1ccc(-c2ccc(C#N)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
CNR1 P21554 2/20 0.50
KDM4E B2RXH2 3/20 0.48
LMNA P02545 5/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 2/20 0.47
MAPK1 P28482 2/20 0.47
KMT2A Q03164 2/20 0.47
SAE1 Q9UBE0 1/20 0.47
UBA2 Q9UBT2 1/20 0.47
POLB P06746 1/20 0.47
PKM P14618 1/20 0.47
RAB9A P51151 1/20 0.47
IL18 Q14116 1/20 0.47
MMP3 P08254 1/20 0.46
PTPN7 P35236 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
NLRP3 Q96P20 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8886444 0.89 CNR1 (0.53) ALDH1A1CNR1KDM4ELMNAMAPT
SCHEMBL4426853 0.83 PPID (0.55) ALDH1A1CNR1KDM4ELMNAMAPT
SCHEMBL8410208 0.82 MAPT (0.52) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL27519540 0.79 ALDH1A1 (0.82) ALDH1A1KDM4ELMNAMAPTMEN1
SCHEMBL7281233 0.79 ALDH1A1 (0.48) ALDH1A1KDM4ELMNAMAPK1MMP3
SCHEMBL14423993 0.79 CNR1 (0.62) ALDH1A1CNR1KDM4ELMNAMAPT
SCHEMBL3929566 0.78 MAPT (0.55) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL8573559 0.78 CNR1 (0.61) ALDH1A1CNR1KDM4ELMNAMAPT
SCHEMBL7389737 0.77 CNR1 (0.60) ALDH1A1CNR1KDM4ELMNAMAPT
SCHEMBL9937346 0.77 ALDH1A1 (0.59) ALDH1A1CNR1KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed