SCHEMBL8409442

SCHEMBL8409442

CC(C)(C)OC(=O)C[C@H](NC(=O)[C@@H]1CCCN2C(=O)CC[C@H](NS(C)(=O)=O)C(=O)N12)C(O)c1nc2cc(Cl)cc(Cl)c2o1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 9/20 0.36
IL1B P01584 2/20 0.35
LCK P06239 10/20 0.34
CASP3 P42574 2/20 0.33
CASP8 Q14790 2/20 0.33
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2216912 1.00 CASP1 (0.36) CASP1IL1BLCKCASP3CASP8
SCHEMBL645660 0.91 CASP1 (0.43) CASP1IL1BLCKCASP3CASP8
SCHEMBL2223156 0.88 CASP1 (0.52) CASP1IL1BLCKCASP3CASP8
SCHEMBL7740043 0.87 LCK (0.35) CASP1IL1BLCKCASP3CASP8
SCHEMBL8412036 0.84 CASP1 (0.38) CASP1IL1BLCKCASP3CASP8
SCHEMBL1410039 0.84 CASP1 (0.38) CASP1IL1BLCKCASP3CASP8
SCHEMBL647783 0.79 CASP1 (0.41) CASP1IL1BLCKCASP3CASP8
SCHEMBL644683 0.79 CASP1 (0.41) CASP1IL1BLCKCASP3CASP8
SCHEMBL13139539 0.79 CASP1 (0.41) CASP1IL1BLCKCASP3CASP8
SCHEMBL646086 0.79 CASP1 (0.60) CASP1IL1BLCKCASP3CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6008217-A AN ENZYME INHIBITOR AGAINST INTERLEUKIN-1B, FOR TREATING APOPTOSIS-MEDIATED DISEASES, INCLUDING INFLAMMATORY DISEASES, AUTOIMMUNE DISEASES, PROLIFERATIVE DISORDERS, INFECTIOUS DISEASES, AND DEGENERATIVE DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 1999-12-28 US disclosed