SCHEMBL841279

SCHEMBL841279

CCCCCNC(=O)N(CCNC(=O)C(CS)CC(C)C)Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 18/20 0.42
MME P08473 10/20 0.42
LTB4R2 Q9NPC1 2/20 0.37
AGTR2 P50052 1/20 0.35
ABCB11 O95342 1/20 0.34
GP6 Q9HCN6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL841138 0.99 AGTR1 (0.42) AGTR1MMELTB4R2AGTR2ABCB11
SCHEMBL840597 0.98 AGTR1 (0.43) AGTR1MMELTB4R2AGTR2ABCB11
SCHEMBL840456 0.95 AGTR1 (0.41) AGTR1MMELTB4R2
SCHEMBL840844 0.92 AGTR1 (0.41) AGTR1MMEAGTR2
SCHEMBL840125 0.91 AGTR1 (0.45) AGTR1MMELTB4R2ABCB11GP6
SCHEMBL841346 0.91 AGTR1 (0.45) AGTR1MMELTB4R2ABCB11GP6
SCHEMBL839995 0.89 AGTR1 (0.39) AGTR1MME
SCHEMBL839522 0.89 AGTR1 (0.38) AGTR1MME
SCHEMBL839949 0.89 AGTR1 (0.41) AGTR1MMELTB4R2ABCB11GP6
SCHEMBL859394 0.89 AGTR1 (0.41) AGTR1MMELTB4R2ABCB11GP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143298-B2 Dual-acting antihypertensive agents THERAVANCE, INC. (US) 2012-03-27 US disclosed