Gitoxigenin

Gitoxigenin

SCHEMBL8417147

C[C@]12CC[C@H](O)C[C@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)[C@@H](C3=CC(=O)OC3)[C@H](O)C[C@]12O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 7/20 1.00
RAB9A P51151 4/20 1.00
CYP2C19 P33261 2/20 1.00
ATP1A1 P05023 7/20 0.74
ATP1B1 P05026 7/20 0.74
ATP1A3 P13637 7/20 0.74
ATP1B2 P14415 7/20 0.74
ATP1A2 P50993 7/20 0.74
ATP1B3 P54709 7/20 0.74
FXYD2 P54710 7/20 0.74
ATP1A4 Q13733 7/20 0.74
SMN1; SMN2 Q16637 4/20 0.74
PAX8 Q06710 3/20 0.74
LMNA P02545 3/20 0.74
NPC1 O15118 3/20 0.74
HIF1A Q16665 2/20 0.74
CYP3A4 P08684 1/20 0.74
TSHR P16473 1/20 0.74
ATP12A P54707 1/20 0.74
SLCO4C1 Q6ZQN7 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gitoxigenin SCHEMBL644087 1.00 TP53 (1.00) TP53RAB9ACYP2C19ATP1A1ATP1B1
Gitoxigenin SCHEMBL3302691 1.00 TP53 (1.00) TP53RAB9ACYP2C19ATP1A1ATP1B1
Gitoxigenin SCHEMBL13338042 1.00 TP53 (1.00) TP53RAB9ACYP2C19ATP1A1ATP1B1
Gitoxigenin SCHEMBL19638184 1.00 TP53 (1.00) TP53RAB9ACYP2C19ATP1A1ATP1B1
Gitoxigenin SCHEMBL3302694 1.00 TP53 (1.00) TP53RAB9ACYP2C19ATP1A1ATP1B1
SCHEMBL14681100 0.88 TP53 (0.79) TP53RAB9ACYP2C19ATP1A1ATP1B1
SCHEMBL4905625 0.88 TP53 (0.84) TP53RAB9ACYP2C19ATP1A1ATP1B1
SCHEMBL17864015 0.88 TP53 (0.84) TP53RAB9ACYP2C19ATP1A1ATP1B1
SCHEMBL11408235 0.87 TP53 (0.77) TP53RAB9ACYP2C19ATP1A1ATP1B1
SCHEMBL21578190 0.87 TP53 (0.77) TP53RAB9ACYP2C19ATP1A1ATP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0941733-A2 Methods of inhibiting leaderless protein export using cardiac glycosides and derivatives The Scripps Research Institute (US) 1999-09-15 EP disclosed
EP-0828497-B1 METHODS OF INHIBITING LEADERLESS PROTEIN EXPORT USING CARDIAC GLYCOSIDES OR AGLYCONES THEREFROM AND DERIVATIVES SCRIPPS RESEARCH INST (US) 1999-09-01 EP disclosed