SCHEMBL8419783

SCHEMBL8419783

CCCCOc1nc(-c2cccc(OC)c2)cc(-c2ccc(S(N)(=O)=O)cc2)c1CO

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.47
CA9 Q16790 10/20 0.47
CA1 P00915 9/20 0.47
CA4 P22748 1/20 0.46
CA5A P35218 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
CA12 O43570 3/20 0.44
TSHR P16473 1/20 0.44
CA7 P43166 1/20 0.44
PTGS2 P35354 3/20 0.43
GCGR P47871 1/20 0.42
CDK2 P24941 2/20 0.42
DHODH Q02127 1/20 0.41
PTGDR Q13258 1/20 0.41
PTGS1 P23219 2/20 0.40
TLR8 Q9NR97 1/20 0.40
SQOR Q9Y6N5 1/20 0.40
CDK1 P06493 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8423418 0.89 PTGS2 (0.44) CA2CA9CA1CA5ACA5B
SCHEMBL8419780 0.87 DHODH (0.41) CA2CA9CA1PTGS2GCGR
SCHEMBL8423494 0.86 PTGS2 (0.42) CA2CA9CA1CA12TSHR
SCHEMBL8419909 0.84 PTGS2 (0.46) CA2CA9CA1CA4CA12
SCHEMBL8419785 0.84 PTGS2 (0.53) PTGS2CDK2PTGS1
SCHEMBL8419437 0.84 PTGS2 (0.53) CA2CA9CA1CA12TSHR
SCHEMBL8421109 0.83 PTGS2 (0.55) CA2CA9CA1CA12TSHR
SCHEMBL8094362 0.82 PTGS2 (0.59) CA2CA9CA1CA4CA5A
SCHEMBL8421302 0.82 PTGS2 (0.44) CA2CA9CA1CA12TSHR
SCHEMBL8421305 0.77 PTGS2 (0.43) CA2CA9CA1CA12TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed