SCHEMBL8420804

SCHEMBL8420804

CS(=O)(=O)c1ccc(-n2nc(-c3ccc(Cl)cc3)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.88

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.88
PTGS1 P23219 4/20 0.67
RARA P10276 1/20 0.57
RARB P10826 1/20 0.57
RARG P13631 1/20 0.57
RXRA P19793 1/20 0.57
ALOX5 P09917 1/20 0.56
CYP2C9 P11712 2/20 0.56
MALT1 Q9UDY8 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8420798 0.95 PTGS2 (0.80) PTGS2PTGS1RARARARBRARG
SCHEMBL8421185 0.95 PTGS2 (0.80) PTGS2PTGS1RARARARBRARG
SCHEMBL8420828 0.95 PTGS2 (0.80) PTGS2PTGS1RARARARBRARG
SCHEMBL8424052 0.95 PTGS2 (0.80) PTGS2PTGS1RARARARBRARG
SCHEMBL8420266 0.94 PTGS2 (0.79) PTGS2PTGS1RARARARBRARG
SCHEMBL8423953 0.94 PTGS2 (0.79) PTGS2PTGS1
SCHEMBL8424042 0.94 PTGS2 (0.83) PTGS2PTGS1RARARARBRARG
SCHEMBL8423360 0.94 PTGS2 (0.79) PTGS2PTGS1RARARARBRARG
SCHEMBL8420040 0.94 PTGS2 (0.79) PTGS2PTGS1RARARARBRARG
SCHEMBL8420755 0.94 PTGS2 (0.79) PTGS2PTGS1RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed
US-5434178-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G.D. SEARLE & CO. (US) 1995-07-18 US disclosed