SCHEMBL8420853

SCHEMBL8420853

CS(=O)(=O)c1ccc(-n2nc(-c3cc(F)ccc3F)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.66
PTGS1 P23219 4/20 0.57
AOC3 Q16853 1/20 0.53
CYP2C9 P11712 1/20 0.49
TGFBR1 P36897 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8422328 0.93 PTGS2 (0.65) PTGS2PTGS1AOC3CYP2C9
SCHEMBL8424109 0.91 PTGS2 (0.66) PTGS2PTGS1AOC3TGFBR1
SCHEMBL8114834 0.89 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL8423870 0.89 PTGS2 (0.79) PTGS2PTGS1AOC3
SCHEMBL8423953 0.89 PTGS2 (0.79) PTGS2PTGS1AOC3
SCHEMBL8420916 0.87 PTGS2 (0.60) PTGS2PTGS1AOC3
SCHEMBL8424144 0.86 PTGS2 (0.65) PTGS2PTGS1AOC3
SCHEMBL8421495 0.86 PTGS2 (0.67) PTGS2PTGS1AOC3CYP2C9
SCHEMBL8421887 0.85 PTGS2 (0.73) PTGS2PTGS1CYP2C9
SCHEMBL8422358 0.85 PTGS2 (0.73) PTGS2PTGS1AOC3CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed
US-5434178-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G.D. SEARLE & CO. (US) 1995-07-18 US disclosed