SCHEMBL8423587

SCHEMBL8423587

C=C1CCCOC12CC[C@H]1[C@@H]3CCC4=CC(=O)CC[C@@H]4[C@H]3CC[C@@]12C

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 6/20 0.60
AR P10275 4/20 0.60
NR3C2 P08235 2/20 0.60
CYP3A4 P08684 3/20 0.56
ABCB11 O95342 3/20 0.56
LMNA P02545 2/20 0.56
CYP2C19 P33261 2/20 0.56
NR3C1 P04150 2/20 0.56
ALDH1A1 P00352 2/20 0.56
SHBG P04278 2/20 0.56
TSHR P16473 1/20 0.56
HIF1A Q16665 1/20 0.56
ESR1 P03372 1/20 0.56
ADRA2A P08913 1/20 0.56
SLC6A4 P31645 1/20 0.56
MAPT P10636 2/20 0.53
CHRM2 P08172 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
CHRM1 P11229 1/20 0.53
TBXA2R P21731 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8423021 0.94 PGR (0.62) PGRARNR3C2CYP3A4ABCB11
SCHEMBL8425076 0.86 PGR (0.64) PGRARNR3C2CYP3A4ABCB11
SCHEMBL8425180 0.85 PGR (0.62) PGRARNR3C2CYP3A4ABCB11
SCHEMBL8423621 0.85 PGR (0.63) PGRARNR3C2CYP3A4ABCB11
SCHEMBL8427213 0.85 PGR (0.54) PGRARNR3C2CYP3A4ABCB11
SCHEMBL8423533 0.82 PGR (0.59) PGRARNR3C2CYP3A4ABCB11
SCHEMBL13062188 0.82 PGR (0.64) PGRARNR3C2CYP3A4ABCB11
SCHEMBL8427388 0.82 PGR (0.58) PGRARNR3C2CYP3A4ABCB11
SCHEMBL11942939 0.80 PGR (0.67) PGRARNR3C2CYP3A4ABCB11
SCHEMBL13160889 0.80 PGR (0.67) PGRARNR3C2CYP3A4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582338-B1 17-Spiromethylene steroids AKZO NOBEL NV (NL) 1999-10-20 EP disclosed
US-5854235-A 17-spiromethylene steroids AKZO NOBEL N.V. (NL) 1998-12-29 US disclosed
US-5712264-A 17-spiromethylene steroids AKZO NOBEL N.V. (NL) 1998-01-27 US disclosed
EP-0582338-A2 17-Spiromethylene steroids Akzo Nobel N.V. (NL) 1994-02-09 EP disclosed