SCHEMBL8424237

SCHEMBL8424237

N=C(Nc1ccc(I)c2ccccc12)Nc1ccc2c3c(cccc13)C=C2

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.33
NPC1 O15118 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
PARP1 P09874 1/20 0.32
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6155027 0.88 KDM4E (0.34) NPC1CYP1A2CYP3A4CYP2D6CYP2C9
Bromide SCHEMBL6154947 0.86 KDM4E (0.33) NPC1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8424098 0.84 SIGMAR1 (0.36) SIGMAR1NPC1CYP1A2CYP3A4CYP2D6
SCHEMBL6155518 0.84 IDO1 (0.44)
SCHEMBL6156264 0.84 KDM4E (0.47) SIGMAR1NPC1CYP1A2CYP3A4CYP2D6
SCHEMBL6155300 0.83 MEN1 (0.36) NPC1RAB9AKDM4EGAA
SCHEMBL6155016 0.83 CDC25B (0.37) SIGMAR1NPC1CYP3A4RAB9AKDM4E
SCHEMBL6719241 0.83 CYP1A2 (0.37) NPC1CYP1A2RAB9AKDM4EGAA
Hydrochloric Acid SCHEMBL8717239 0.82 CYP1A2 (0.36) CYP1A2KDM4EGAA
SCHEMBL8424140 0.80 KDM4E (0.35) CYP1A2CYP2C19KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0584088-B1 SUBSTITUTED GUANIDINES AND DERIVATIVES THEREOF AS MODULATORS OF NEUROTRANSMITTER RELEASE AND NOVEL METHODOLOGY FOR IDENTIFYING NEUROTRANSMITTER RELEASE BLOCKERS CAMBRIDGE NEUROSCIENCE RES (US) 1999-10-27 EP claimed