SCHEMBL8424939

SCHEMBL8424939

C=CC(C)(O)CC/C=C(/C)CO

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 4/20 0.68
BTN3A1 O00481 9/20 0.38
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR2 P34972 1/20 0.32
HIF1A Q16665 2/20 0.31
EPAS1 Q99814 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3499478 1.00 ALOX15 (0.68) ALOX15BTN3A1MEN1CYP3A4KMT2A
SCHEMBL28423346 1.00 ALOX15 (0.68) ALOX15BTN3A1MEN1CYP3A4KMT2A
SCHEMBL3499480 1.00 ALOX15 (0.68) ALOX15BTN3A1MEN1CYP3A4KMT2A
SCHEMBL9421358 0.93 ALOX15 (0.78) ALOX15BTN3A1MEN1CYP3A4KMT2A
SCHEMBL9421355 0.93 ALOX15 (0.78) ALOX15BTN3A1MEN1CYP3A4KMT2A
SCHEMBL164898 0.86 ALOX15 (0.70) ALOX15MEN1CYP3A4KMT2AHIF1A
SCHEMBL296693 0.86 ALOX15 (0.70) ALOX15MEN1CYP3A4KMT2AHIF1A
SCHEMBL31678342 0.86 ALOX15 (0.70) ALOX15MEN1CYP3A4KMT2AHIF1A
SCHEMBL296694 0.86 ALOX15 (0.70) ALOX15MEN1CYP3A4KMT2AHIF1A
SCHEMBL1325095 0.82 ALOX15 (0.68) ALOX15MEN1CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2718309-B1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS KEYGENE NV (NL) 2018-04-04 EP disclosed
US-20170247713-A1 TRICHOME-SPECIFIC TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS KEYGENE N.V. (NL) 2017-08-31 US disclosed
US-9598473-B2 Trichome-specific transcription factor modulating terpene biosynthesis KEYGENE N.V. (NL) 2017-03-21 US disclosed
US-20140173771-A1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS Stichting Techno. Topinstituut Groene Genetica (Foundation Techno. top Institute Green Genetics) 2014-06-19 US disclosed
EP-2718309-A1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS Stichting Technologisch Topinstituut Groene Genetica (Foundation Technological Top Institute Green Genetics) (NL) 2014-04-16 EP disclosed
WO-2012169893-A1 TRANSCRIPTION FACTOR MODULATING TERPENE BIOSYNTHESIS STICHTING TECHNOLOGISCH TOPINSTITUUT GROENE GENETICA (FOUNDATION TECHNOLOGICAL TOP INSTITUTE GREEN GENETICS) (NL) 2012-12-13 WO disclosed
US-5985618-A ENZYMATICALLY HYDROLYZING CIST-BROCADES, N.V. (NL) 1999-11-16 US disclosed
EP-0416713-B2 Process for obtaining aroma components and aromas from their precursors of a glycosidic nature, and aroma components and aromas thereby obtained DSM NV (NL) 1999-06-23 EP disclosed
WO-1991003174-A1 PROCESS FOR OBTAINING AROMA COMPONENTS AND AROMAS FROM THEIR PRECURSORS OF A GLYCOSIDIC NATURE, AND AROMA COMPONENTS AND AROMAS THEREBY OBTAINED GIST-BROCADES N.V. (NL) 1991-03-21 WO disclosed
EP-0416713-A1 Process for obtaining aroma components and aromas from their precursors of a glycosidic nature, and aroma components and aromas thereby obtained GIST-BROCADES N.V. (NL) 1991-03-13 EP disclosed