SCHEMBL8425919

SCHEMBL8425919

N=C(Nc1ccc(C2CC2)cc1)Nc1ccc2c3c(cccc13)C=C2

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
IDO1 P14902 2/20 0.30
NAMPT P43490 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
DEGS1 O15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6727607 0.94 HDAC3 (0.38) HDAC3HDAC11HDAC8HDAC6RAB9A
Hydrochloric Acid SCHEMBL8711917 0.93 HDAC3 (0.38) HDAC3HDAC11HDAC8HDAC6RAB9A
SCHEMBL6155027 0.82 KDM4E (0.34) RAB9AKMT2AKDM4EMAPTLMNA
SCHEMBL8424104 0.82 HDAC3 (0.33) HDAC3HDAC11HDAC8HDAC6
SCHEMBL6716804 0.82 TRPV1 (0.40) RAB9AKMT2AKDM4EMAPTLMNA
Bromide SCHEMBL6154947 0.81 KDM4E (0.33) RAB9AKMT2AKDM4EMAPTLMNA
SCHEMBL6720772 0.79 TRPV1 (0.44) RAB9AKMT2AMAPT
SCHEMBL6156272 0.79 GAA (0.48) RAB9AKMT2AKDM4EMAPTLMNA
SCHEMBL6720829 0.79 RAB9A (0.43) RAB9AKMT2AKDM4EMAPTLMNA
SCHEMBL6720912 0.79 HTR2C (0.42) RAB9AKMT2AKDM4EMAPTIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0584088-B1 SUBSTITUTED GUANIDINES AND DERIVATIVES THEREOF AS MODULATORS OF NEUROTRANSMITTER RELEASE AND NOVEL METHODOLOGY FOR IDENTIFYING NEUROTRANSMITTER RELEASE BLOCKERS CAMBRIDGE NEUROSCIENCE RES (US) 1999-10-27 EP claimed