SCHEMBL8427620

SCHEMBL8427620

CC(C=O)c1cnccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.37
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSP90AA1 P07900 1/20 0.33
NAPRT Q6XQN6 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
ATM Q13315 1/20 0.33
ADORA3 P0DMS8 1/20 0.32
TSHR P16473 1/20 0.32
MC4R P32245 1/20 0.32
ADRA1A P35348 1/20 0.32
MC3R P41968 1/20 0.32
VNN1 O95497 3/20 0.32
FFAR2 O15552 1/20 0.32
HPGDS O60760 1/20 0.32
CYP2D6 P10635 1/20 0.31
CHRM1 P11229 1/20 0.31
HRH1 P35367 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL294331 0.81 KDM4E (0.35) LMNAKDM4EALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL21284664 0.79 KDM4E (0.34) LMNAKDM4EALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL13397712 0.79 KDM4E (0.34) LMNAKDM4EALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL2558175 0.78 HSP90AA1 (0.36) LMNAKDM4EHSP90AA1NAPRTHCAR2
SCHEMBL839685 0.76
SCHEMBL1919145 0.75 KDM4E (0.33) LMNAKDM4EHSP90AA1NAPRTHCAR2
SCHEMBL29738290 0.75
SCHEMBL681871 0.75
SCHEMBL8475264 0.75 KDM4E (0.35) LMNAKDM4EALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL11842818 0.75 ATM (0.39) KDM4EHSP90AA1NAPRTHCAR2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513020-B KDM1A inhibitors for the treatment of diseases 伊美格生物科学公司 2024-02-23 CN disclosed
CN-1980578-B Encapsulated hydrophilic compounds FIRMENICH & CIE 2010-10-13 CN disclosed
CN-1997649-B Inhibitors of histone deacetylase METHYLGENE INC 2010-08-11 CN disclosed
CN-100436445-C Pyrazole derivative DAIICHI SEIYAKU CO (JP) 2008-11-26 CN disclosed
CN-101001852-A Pyrazole derivatives DAIICHI SEIYAKU CO (JP) 2007-07-18 CN disclosed
CN-1997649-A Inhibitors of histone deacetylase METHYLGENE INC (CA) 2007-07-11 CN disclosed
CN-1980578-A Encapsulated hydrophilic compounds FIRMENICH & CIE (CH) 2007-06-13 CN disclosed
CN-1902191-A Amidopyrazole derivative DAIICHI SEIYAKU CO (JP) 2007-01-24 CN disclosed
CN-1759110-A Pyrazole derivatives DAIICHI SEIYAKU CO (JP) 2006-04-12 CN disclosed
US-5973156-A Piperidine and tetrahydropyridine derivatives MERCK SHARP & DOME LTD. (GB) 1999-10-26 US disclosed
EP-0861245-A1 PIPERIDINE AND TETRAHYDROPYRIDINE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1998-09-02 EP disclosed
WO-1997019073-A1 PIPERIDINE AND TETRAHYDROPYRIDINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1997-05-29 WO disclosed
US-3941781-A Preparation of 3-alkylthiomethyl cephalosporins ELI LILLY AND COMPANY (US) 1976-03-02 US disclosed