SCHEMBL8427633

SCHEMBL8427633

CCOC(=O)Nc1ccc(N2N=C(C)CC2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
MAPT P10636 5/20 0.54
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
TDP1 Q9NUW8 4/20 0.54
LMNA P02545 2/20 0.54
HTT P42858 1/20 0.54
KDM4E B2RXH2 5/20 0.52
GAA P10253 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
CYP1A2 P05177 1/20 0.52
CHRM2 P08172 1/20 0.52
CYP3A4 P08684 1/20 0.52
CHRM1 P11229 1/20 0.52
TSHR P16473 1/20 0.52
PTGS1 P23219 1/20 0.52
DRD3 P35462 1/20 0.52
RECQL P46063 2/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8424148 0.88 APP (0.58) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL6945778 0.84 MAPT (0.56) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL8020214 0.83 KMT2A (0.66) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL8423947 0.82 KMT2A (0.60) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL4661824 0.81 MAPT (0.61) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL11870457 0.78 MEN1 (0.67) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL4663160 0.77 MAPT (0.62) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL13122202 0.77 NPC1 (0.59) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL8428074 0.77 GAA (0.59) ALDH1A1MAPTMEN1KMT2ATDP1
SCHEMBL8427533 0.77 MAPT (0.65) ALDH1A1MAPTMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869516-A 4-(arylaminomethylene)-2,4-dihydro-3-pyrazolones MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-02-09 US disclosed