SCHEMBL8430475

SCHEMBL8430475

C=CCC(O)CCC[C@@H](C(=O)O)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
POLB P06746 4/20 0.57
KDM4E B2RXH2 1/20 0.57
TP53 P04637 1/20 0.57
GLA P06280 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
HPGD P15428 1/20 0.57
ALOX12 P18054 1/20 0.57
NFKB1 P19838 1/20 0.57
APEX1 P27695 1/20 0.57
MAPK1 P28482 1/20 0.57
HSD17B10 Q99714 1/20 0.57
GAA P10253 2/20 0.51
DNMT1 P26358 5/20 0.44
HIF1A Q16665 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
KMT2A Q03164 3/20 0.42
PKM P14618 2/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL84217 0.83 ALDH1A1 (0.62) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL3721573 0.83 ALDH1A1 (0.62) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL8432059 0.80 POLB (0.64) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL10492337 0.79 ALDH1A1 (0.68) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL7349189 0.77 ALDH1A1 (0.64) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL7349201 0.77 ALDH1A1 (0.64) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL10492333 0.77 ALDH1A1 (0.64) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL9741723 0.76 ALDH1A1 (0.82) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL5828001 0.76 ALDH1A1 (0.68) ALDH1A1POLBKDM4ETP53GLA
SCHEMBL5828004 0.76 ALDH1A1 (0.68) ALDH1A1POLBKDM4ETP53GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859239-A Mercaptoalkanoylamino and acylmercaptoalkanoylamino benzoxazepines and benzothiazepines E. R. SQUIBB & SONS, INC. (US) 1999-01-12 US disclosed
US-5856476-A Processes for preparing azepiones useful as intermediates in the preparation of inhibitors of angiotensin converting enzyme and neutral endopeptidase E. R. SQUIBBS & SONS, INC. (US) 1999-01-05 US disclosed
US-5856477-A HYPOTENSIVE AGENTS; CONGESTIVE HEART FAILURE E. R. SQUIBB & SONS, INC. (US) 1999-01-05 US disclosed
US-5723602-A ANGIOTENSIN CONVERTING ENZYME AND ENDOPEPTIDASE INHIBITORS, CARDIOVASCULAR DISORDERS E. R. SQUIBB & SONS, INC. (US) 1998-03-03 US disclosed
US-5723457-A COMPOUMDS FOR CARDIOVASCULAR DISORDERS AND INHIBITORS OF ANGIOTENSIN CONVERTING ENZYMES E. R. SQUIBB & SONS, INC. (US) 1998-03-03 US disclosed
US-5654294-A CARDIOVASCULAR DISORDERS BRISTOL-MYERS SQUIBB (US) 1997-08-05 US disclosed
US-5646276-A ANGIOTENSIN CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE INHIBITORS; CARDIOVASCULAR DISORDERS BRISTOL-MYERS SQUIBB CO. (US) 1997-07-08 US disclosed
US-5552397-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-09-03 US disclosed