SCHEMBL8432503

SCHEMBL8432503

NCCc1csc2ccc(C3CCC3)cc12

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.52
HTR5A P47898 1/20 0.43
CYP2A6 P11509 3/20 0.41
MTNR1A P48039 4/20 0.40
MTNR1B P49286 3/20 0.40
HTR2A P28223 2/20 0.37
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
EPHX1 P07099 1/20 0.35
NUDT1 P36639 1/20 0.35
BACE1 P56817 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431855 0.94 HTR1D (0.48) HTR1DHTR5ACYP2A6MTNR1AMTNR1B
SCHEMBL27492816 0.79 MTNR1A (0.43) HTR1DMTNR1AMTNR1BEPHX1HRH3
SCHEMBL27468521 0.77 MTNR1A (0.63) MTNR1AMTNR1B
SCHEMBL27508400 0.76 MTNR1A (0.67) MTNR1AMTNR1B
SCHEMBL27450736 0.76 MTNR1A (0.65) MTNR1AMTNR1B
SCHEMBL8591649 0.75 CYP2A6 (0.50) HTR5ACYP2A6MTNR1AMTNR1B
SCHEMBL27468028 0.75 MTNR1A (0.59) MTNR1AMTNR1BSMN1; SMN2
SCHEMBL27449304 0.72 MTNR1A (0.67) MTNR1AMTNR1B
SCHEMBL4324624 0.72 CYP2A6 (0.75) HTR5ACYP2A6HTR2AEPHX1SMN1; SMN2
SCHEMBL8586692 0.72 HTR2C (0.49) HTR1DHTR5ACYP2A6MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721938-B1 Alkyl(hetero)cyclic compounds, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1999-12-08 EP disclosed
EP-0721938-A1 Alkyl(hetero)cyclic compounds, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-07-17 EP disclosed