SCHEMBL8433686

SCHEMBL8433686

CC(C)[C@H](N)C(O)c1noc(Cc2ccsc2)n1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
IDH1 O75874 1/20 0.31
SLC1A3 P43003 2/20 0.30
SLC1A2 P43004 2/20 0.30
SLC1A1 P43005 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8435682 0.99 PTGS1 (0.33) PTGS1PTGS2IDH1
SCHEMBL8433420 0.82 IDH1 (0.42) IDH1
Hydrochloric Acid SCHEMBL8434597 0.81 IDH1 (0.41) IDH1
SCHEMBL8438545 0.78 SMN1; SMN2 (0.49)
Hydrochloric Acid SCHEMBL8437554 0.77 SMN1; SMN2 (0.48)
Hydrochloric Acid SCHEMBL8495697 0.76 RAB9A (0.44) IDH1
SCHEMBL8432982 0.74 TAAR1 (0.45)
SCHEMBL8434690 0.74 PRSS1 (0.47)
Hydrochloric Acid SCHEMBL8435752 0.74 TAAR1 (0.44)
Hydrochloric Acid SCHEMBL8435334 0.73 IDH1 (0.33) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874585-A TREATMENT AND/OR PREVENTION OF ELASTASE-MEDIATED PROBLEMS SUCH AS ARTHRITIS, PERIODONTAL DISEASE, GLOMERULONEPHRITIS, DERMATITIS, PSORIASIS, CYSTIC FIBROSIS, CHRONIC BRONCHITIS, ALZHEIMER'S DISEASE CORTECH, INC. (US) 1999-02-23 US disclosed