SCHEMBL8436141

SCHEMBL8436141

O=C(O)c1ccc(C(=O)c2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 9/20 1.00
TSHR P16473 3/20 0.76
EPHX2 P34913 1/20 0.56
ALOX15 P16050 2/20 0.52
TP53 P04637 1/20 0.50
VCAM1 P19320 1/20 0.49
TTR P02766 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6322177 0.89 SRD5A2 (0.79) SRD5A2TSHRVCAM1
SCHEMBL333237 0.88 SRD5A2 (0.78) SRD5A2TSHRALOX15VCAM1
SCHEMBL8352471 0.87 TSHR (1.00) SRD5A2TSHREPHX2ALOX15TTR
SCHEMBL29353637 0.87 TSHR (1.00) SRD5A2TSHREPHX2ALOX15TTR
SCHEMBL371998 0.87 TSHR (1.00) SRD5A2TSHREPHX2ALOX15TTR
SCHEMBL4052954 0.86 SRD5A2 (0.76) SRD5A2TSHREPHX2ALOX15VCAM1
SCHEMBL9225999 0.85 TSHR (0.95) SRD5A2TSHREPHX2ALOX15TTR
SCHEMBL4847012 0.85 TSHR (0.95) SRD5A2TSHREPHX2ALOX15TTR
SCHEMBL10603908 0.85 TSHR (0.95) SRD5A2TSHREPHX2ALOX15TTR
Hydrochloric Acid SCHEMBL11133785 0.85 TSHR (0.95) SRD5A2TSHREPHX2ALOX15TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998433-A THERAPY FOR HYPERLIPIDEMIA; ATHEROSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-12-07 US disclosed
CN-1160403-A Substd. heterobicyclic alkyl amines and their use as squalene oxide cyclase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-09-24 CN disclosed
EP-0785939-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-30 EP disclosed
WO-1996011201-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-18 WO disclosed