SCHEMBL8437847

SCHEMBL8437847

Cc1nc(CC(C)C(N)CO)no1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8434263 0.98
SCHEMBL8435799 0.80 HDAC4 (0.31)
SCHEMBL8434579 0.80 HDAC4 (0.39)
Hydrochloric Acid SCHEMBL8438947 0.78 HDAC4 (0.38)
Hydrochloric Acid SCHEMBL8433618 0.78 HDAC4 (0.30)
SCHEMBL8433805 0.75 NOTUM (0.57)
Hydrochloric Acid SCHEMBL8437873 0.74 NOTUM (0.56)
SCHEMBL1913015 0.74 GCGR (0.35)
SCHEMBL8433601 0.73 ALDH1A1 (0.35)
SCHEMBL8433423 0.73 TDP1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874585-A TREATMENT AND/OR PREVENTION OF ELASTASE-MEDIATED PROBLEMS SUCH AS ARTHRITIS, PERIODONTAL DISEASE, GLOMERULONEPHRITIS, DERMATITIS, PSORIASIS, CYSTIC FIBROSIS, CHRONIC BRONCHITIS, ALZHEIMER'S DISEASE CORTECH, INC. (US) 1999-02-23 US disclosed