SCHEMBL8440232

SCHEMBL8440232

COC(=O)c1ccc2c(C(=O)c3ccc4ccccc4c3)c(C(=O)OC)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.52
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48
ALDH1A1 P00352 7/20 0.47
KDM4E B2RXH2 5/20 0.47
PLAU P00749 2/20 0.47
ALOX12 P18054 1/20 0.47
HPGD P15428 4/20 0.47
MAPT P10636 3/20 0.47
GLA P06280 2/20 0.47
GAA P10253 2/20 0.47
ATM Q13315 2/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
HSD17B10 Q99714 1/20 0.47
LMNA P02545 1/20 0.46
PTPN11 Q06124 2/20 0.45
KIF11 P52732 1/20 0.45
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8442119 0.90 LCK (0.54) LCKSLC6A3ALDH1A1KDM4EPLAU
SCHEMBL9002749 0.87 LCK (0.48) LCKALDH1A1KDM4EPLAUALOX12
SCHEMBL7558686 0.84 KDM4E (0.49) ALDH1A1KDM4EPLAUHPGDMAPT
SCHEMBL1003761 0.82 KDM4E (0.62) LCKSLC6A2SLC6A4SLC6A3ALDH1A1
Hydrochloric Acid SCHEMBL15414839 0.81 KDM4E (0.60) LCKSLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL27607386 0.79 ALDH1A1 (0.67) LCKALDH1A1KDM4EPLAUHPGD
SCHEMBL30213808 0.78 LCK (0.58) LCKSLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL69179 0.78 LCK (0.58) LCKSLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL28514499 0.78 KDM4E (0.57) LCKSLC6A2SLC6A4SLC6A3ALDH1A1
Boric Acid SCHEMBL28499454 0.78 KDM4E (0.57) LCKSLC6A2SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713501-B1 NAPHTHALENEDICARBOXYLIC ACID CONTAINING POLYMERS HAVING REDUCED FLUORESCENCE EASTMAN CHEM CO (US) 1997-04-23 EP claimed
EP-0731783-A1 NAPHTHALENE DICARBOXYLIC ACIDS AND ESTERS SUBSTITUTED WITH AROYL GROUPS EASTMAN CHEMICAL COMPANY (US) 1996-09-18 EP claimed
EP-0713501-A1 NAPHTHALENEDICARBOXYLIC ACID CONTAINING POLYMER COMPOSITIONS HAVING REDUCED FLUORESCENCE EASTMAN CHEM CO (US) 1996-05-29 EP claimed
WO-1995015304-A1 NAPHTHALENE DICARBOXYLIC ACIDS AND ESTERS SUBSTITUTED WITH AROYL GROUPS EASTMAN CHEMICAL COMPANY (US) 1995-06-08 WO claimed
US-5393862-A Heat resistance; high glass transition temperature, gas barrier EASTMAN CHEMICAL COMPANY (US) 1995-02-28 US claimed
WO-1995004768-A1 NAPHTHALENEDICARBOXYLIC ACID CONTAINING POLYMER COMPOSITIONS HAVING REDUCED FLUORESCENCE EASTMAN CHEMICAL COMPANY (US) 1995-02-16 WO claimed
US-5352761-A Incorporated into polyesters for reduced fluorescence EASTMAN CHEMICAL COMPANY (US) 1994-10-04 US claimed
US-5310857-A Packaging materials EASTMAN CHEMICAL COMPANY (US) 1994-05-10 US claimed
US-5919403-A POLYESTERS EASTMAN CHEMICAL COMPANY (US) 1999-07-06 US disclosed
EP-0868488-A1 NAPHTHALENEDICARBOXYLATE CONTAINING POLYESTER BLEND COMPOSITIONS HAVING REDUCED FLUORESCENCE EASTMAN CHEMICAL COMPANY (US) 1998-10-07 EP disclosed
EP-0868465-A1 POLYMERIC FLUORESCENCE QUENCHING COMPOUNDS AND THEIR USE EASTMAN CHEMICAL COMPANY (US) 1998-10-07 EP disclosed
US-5705600-A MELT BLENDING A POLYESTER AND POLYAMIDE WITH FLUORESCENCE QUENCHING COMPOUND EASTMAN CHEMICAL COMPANY (US) 1998-01-06 US disclosed
WO-1997023568-A1 NAPHTHALENEDICARBOXYLATE CONTAINING POLYESTER BLEND COMPOSITIONS HAVING REDUCED FLUORESCENCE EASTMAN CHEMICAL COMPANY (US) 1997-07-03 WO disclosed
WO-1997023569-A1 POLYESTER/NAPHTHALENEDICARBOXYLIC ACID-CONTAINING POLYMER BLENDS DISPLAYING REDUCED FLUORESCENCE EASTMAN CHEMICAL COMPANY (US) 1997-07-03 WO disclosed
US-5391702-A Melt blending with a fluorescence-quenching aromatic ketone or aromatic alcohol and forming EASTMAN CHEMICAL COMPANY (US) 1995-02-21 US disclosed
US-5391330-A Melt blending aromatic ketone or naphthol compounds EASTMAN CHEMICAL COMPANY (US) 1995-02-21 US disclosed
WO-1995004768-A1 NAPHTHALENEDICARBOXYLIC ACID CONTAINING POLYMER COMPOSITIONS HAVING REDUCED FLUORESCENCE EASTMAN CHEMICAL COMPANY (US) 1995-02-16 WO disclosed
WO-1995004777-A1 A PROCESS FOR PREPARING NAPHTHALENEDICARBOXYLIC ACID CONTAINING POLYMER BLENDS HAVING REDUCED FLUORESCENCE EASTMAN CHEMICAL COMPANY (US) 1995-02-16 WO disclosed
US-5352761-A Incorporated into polyesters for reduced fluorescence EASTMAN CHEMICAL COMPANY (US) 1994-10-04 US disclosed
US-5310857-A Packaging materials EASTMAN CHEMICAL COMPANY (US) 1994-05-10 US disclosed