SCHEMBL8441650

SCHEMBL8441650

CC(O)c1ccc(Cl)c(Cl)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.46
CYP3A4 P08684 2/20 0.42
MAPK1 P28482 1/20 0.42
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
NFKB1 P19838 1/20 0.39
PNMT P11086 1/20 0.39
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
AHR P35869 2/20 0.32
TDP1 Q9NUW8 1/20 0.31
DRD2 P14416 2/20 0.31
DRD3 P35462 2/20 0.31
TSHR P16473 1/20 0.31
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17858501 0.80 PDE2A (0.46) PDE2ACYP3A4MAPK1CYP1A2CYP2D6
SCHEMBL9806515 0.80 PDE2A (0.42) PDE2ACYP3A4CYP1A2CYP2D6NFKB1
SCHEMBL14373062 0.80 CYP3A4 (0.41) PDE2ACYP3A4MAPK1CYP1A2CYP2D6
SCHEMBL7546175 0.79 CYP1A2 (0.63) PDE2ACYP3A4CYP1A2CYP2D6NFKB1
SCHEMBL12061470 0.79 PDE2A (0.40) PDE2ACYP3A4LMNAALDH1A1
SCHEMBL11501879 0.78 CYP3A4 (0.40) PDE2ACYP3A4MAPK1CYP1A2CYP2D6
SCHEMBL17069821 0.77 PDE2A (0.39) PDE2ANOTUM
SCHEMBL17553337 0.76 CYP3A4 (0.39) CYP3A4MAPK1CYP1A2CYP2D6NFKB1
SCHEMBL8440315 0.76 P2RX7 (0.46) CYP3A4MAPK1CYP1A2CYP2D6NFKB1
SCHEMBL16958286 0.76 CYP3A4 (0.39) CYP3A4MAPK1CYP1A2CYP2D6NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604857-B1 Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO (JP) 1999-03-17 EP disclosed
US-5495012-A Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO., LTD. (JP) 1996-02-27 US disclosed
US-5424446-A Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO., LTD. (JP) 1995-06-13 US disclosed
EP-0604857-A1 Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor TANABE SEIYAKU CO., LTD. (JP) 1994-07-06 EP disclosed