SCHEMBL8444075

SCHEMBL8444075

COC(=O)c1cccc(-c2cc(O)cc(O)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.60
CA12 O43570 4/20 0.58
CA9 Q16790 4/20 0.58
CA1 P00915 3/20 0.58
CA2 P00918 3/20 0.58
CA7 P43166 2/20 0.58
CA14 Q9ULX7 2/20 0.58
GABRG2 P18507 1/20 0.54
GABRB3 P28472 1/20 0.54
GABRA5 P31644 1/20 0.54
GABRA3 P34903 1/20 0.54
PLAU P00749 2/20 0.52
CDK8 P49336 1/20 0.52
TSHR P16473 1/20 0.50
LOXL2 Q9Y4K0 1/20 0.50
EGFR P00533 1/20 0.49
CYP4F2 P78329 1/20 0.49
CYP4A11 Q02928 1/20 0.49
XDH P47989 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6434807 0.91 ERN1 (0.61) ERN1CA12CA9CA1CA2
SCHEMBL14880009 0.89 ERN1 (0.59) ERN1CA12CA9CA1CA2
SCHEMBL67941 0.89 CA12 (0.68) ERN1CA12CA9CA1CA2
SCHEMBL27715902 0.87 CA12 (0.71) ERN1CA12CA9CA1CA2
SCHEMBL1661764 0.86 CA12 (0.66) ERN1CA12CA9CA1CA2
SCHEMBL30443216 0.86 CA12 (0.66) ERN1CA12CA9CA1CA2
SCHEMBL29410906 0.84 TSHR (0.67) ERN1CA12CA9CA1CA2
SCHEMBL1221576 0.84 TSHR (0.67) ERN1CA12CA9CA1CA2
SCHEMBL8442658 0.83 CA12 (0.57) ERN1CA12CA9CA1CA2
SCHEMBL731372 0.83 CA12 (0.63) ERN1CA12CA9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968985-A INHIBITORS OF SODIUM ION/HYDROGEN ION EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-19 US disclosed
EP-0773927-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-21 EP disclosed
WO-1996004241-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-15 WO disclosed