SCHEMBL8445699

SCHEMBL8445699

CCCCOC(=O)Nc1nc(C(=NOC(c2ccccc2)(c2ccccc2)c2ccccc2)C(=O)O)cs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.47
MAPK1 P28482 1/20 0.47
ALDH1A1 P00352 3/20 0.46
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
NFKB1 P19838 1/20 0.46
STAT1 P42224 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
GAA P10253 5/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GLS O94925 1/20 0.40
MAPT P10636 4/20 0.40
MEN1 O00255 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8445698 1.00 TSHR (0.47) TSHRMAPK1ALDH1A1RAB9ANPC1
SCHEMBL2877170 0.83 GAA (0.43) MAPK1ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL2877169 0.83 GAA (0.43) MAPK1ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL2877172 0.83 GAA (0.43) MAPK1ALDH1A1RAB9ANPC1SMN1; SMN2
Potassium SCHEMBL8627342 0.82 GAA (0.43) MAPK1ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL8627333 0.82 GAA (0.43) MAPK1ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL8575344 0.81 HDAC3 (0.39) MAPK1ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL12333890 0.81 MAPT (0.48) MAPK1RAB9ANPC1SMN1; SMN2GAA
SCHEMBL19426145 0.79 TSHR (0.42) TSHRMAPK1ALDH1A1RAB9ANPC1
SCHEMBL2450269 0.78 MAPT (0.45) MAPK1RAB9ANPC1SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0594263-B1 INTERMEDIATES FOR THE PREPARATION OF THIOALKYLTHIO CEPHALOSPORIN DERIVATIVES SHIONOGI & CO (JP) 1999-06-09 EP disclosed
EP-0594263-A1 Thioalkylthio cephalosporin derivatives and intermediates SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1994-04-27 EP disclosed