SCHEMBL8446355

SCHEMBL8446355

CCC[C@@H]1CCCc2c1cnn2-c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.66
TMEM97 Q5BJF2 1/20 0.66
DHODH Q02127 6/20 0.45
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
NR4A3 Q92570 1/20 0.38
FPR1 P21462 1/20 0.38
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8443689 0.89 SIGMAR1 (0.62) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL956196 0.88 SIGMAR1 (0.67) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL3455799 0.88 SIGMAR1 (0.67) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL3380893 0.88 SIGMAR1 (0.67) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL9277437 0.88 SIGMAR1 (0.67) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL3377712 0.87 SIGMAR1 (0.66) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL955672 0.87 SIGMAR1 (0.66) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL3455854 0.87 SIGMAR1 (0.66) SIGMAR1TMEM97DHODHKEAP1NFE2L2
SCHEMBL953780 0.84 SIGMAR1 (0.83) SIGMAR1TMEM97DHODH
SCHEMBL958221 0.84 SIGMAR1 (0.83) SIGMAR1TMEM97DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010066829-A1 PROCESS FOR OBTAINING ENANTIOMERICALLY ENRICHED PYRAZOLE DERIVATIVES LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2010-06-17 WO disclosed
EP-2196458-A1 Process for obtaining enantiomerically enriched pyrazole derivatives Laboratorios Del. Dr. Esteve, S.A. (ES) 2010-06-16 EP disclosed