SCHEMBL845253

SCHEMBL845253

Cc1cc(CC(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4C(=O)CN(C)C)cc3)cc2)on1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
VHL P40337 2/20 0.43
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.38
CCNE1 P24864 2/20 0.38
CDK2 P24941 2/20 0.38
GSK3B P49841 1/20 0.38
LMNA P02545 1/20 0.37
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
KMT2A Q03164 3/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13272388 1.00 VHL (0.43) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL845390 0.94 VHL (0.48) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL844965 0.89 VHL (0.44) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL844966 0.89 VHL (0.44) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL13272504 0.89 VHL (0.44) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL845607 0.88 VHL (0.43) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL844964 0.88 CNR2 (0.44) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL845719 0.87 VHL (0.41) VHLALDH1A1TSHRCCNE1CDK2
SCHEMBL844902 0.85 ALDH1A1 (0.47) ALDH1A1TSHRLMNAHCRTR1HCRTR2
SCHEMBL13272496 0.84 VHL (0.40) VHLALDH1A1TSHRCCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
EP-1893573-B1 INHIBITORS OF HCV REPLICATION BRISTOL MYERS SQUIBB CO (US) 2010-07-21 EP disclosed