SCHEMBL8456922

SCHEMBL8456922

COc1ccccc1C(CO)COCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
POLB P06746 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CA1 P00915 5/20 0.44
CA2 P00918 3/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
AGTR1 P30556 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
ACHE P22303 1/20 0.41
TSHR P16473 1/20 0.41
ALOX5 P09917 1/20 0.41
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
SGMS2 Q8NHU3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8148897 1.00 HTT (0.47) HTTL3MBTL1POLBNPSR1CA1
SCHEMBL8156476 0.85 HTT (0.43) HTTL3MBTL1POLBNPSR1CA1
SCHEMBL9220799 0.75 POLB (0.51) HTTL3MBTL1POLBNPSR1CA1
SCHEMBL29127924 0.75 CA1 (0.52) L3MBTL1CA1CA2KMT2AALDH1A1
SCHEMBL28570763 0.74 POLB (0.50) HTTL3MBTL1POLBNPSR1CA1
SCHEMBL28570761 0.74 POLB (0.50) HTTL3MBTL1POLBNPSR1CA1
SCHEMBL13332285 0.73 TACR1 (0.40) HTTCA1CA2CA7CA9
SCHEMBL16737506 0.73 TACR1 (0.40) HTTCA1CA2CA7CA9
SCHEMBL16737507 0.73 TACR1 (0.40) HTTCA1CA2CA7CA9
SCHEMBL10564876 0.72 KMT2A (0.51) HTTPOLBCA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906315-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1999-04-07 EP disclosed
WO-1997049710-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1997-12-31 WO disclosed