SCHEMBL846098

SCHEMBL846098

O=C(Nc1cnc2ccccc2c1Cl)Oc1ccc2c(ccn2C2CCCCC2)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 3/20 0.41
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 3/20 0.38
TP53 P04637 2/20 0.38
FAAH O00519 1/20 0.37
EPHX1 P07099 1/20 0.37
MALT1 Q9UDY8 2/20 0.36
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
AURKA O14965 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
MAPT P10636 3/20 0.34
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
P2RX7 Q99572 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL846696 0.85 BCHE (0.43) ALDH1A1TP53GAAKMT2AMAPT
SCHEMBL846996 0.83 KDM4E (0.42) KDM4CKDM4EALDH1A1TP53FAAH
SCHEMBL844641 0.83 HDAC1 (0.41) KDM4CKDM4EALDH1A1MALT1KMT2A
SCHEMBL844640 0.83 HDAC1 (0.41) KDM4CKDM4EALDH1A1MALT1KMT2A
SCHEMBL848239 0.82 RAB9A (0.47) KDM4CKDM4EALDH1A1TP53FAAH
SCHEMBL2708377 0.69 NPC1 (0.53) KDM4EALDH1A1MAPTNPC1RAB9A
SCHEMBL846901 0.68 TRPV1 (0.61) KDM4EALDH1A1TP53MAPTNPC1
SCHEMBL846141 0.67 MAPT (0.42) ALDH1A1TP53GAAKMT2AMAPT
SCHEMBL846808 0.67 KDM4E (0.45) KDM4EALDH1A1TP53GAAKMT2A
SCHEMBL846572 0.66 HDAC1 (0.44) ALDH1A1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603883-B1 QUINOLINE-DERIVED AMIDE MODULATORS OF VANILLOID VR1 RECEPTOR JANSSEN PHARMACEUTICA NV (BE) 2012-03-28 EP claimed