SCHEMBL846259

SCHEMBL846259

CNc1cc2c(cn1)CC1(C2)C(=O)Nc2ncccc21

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CALCA P06881 2/20 0.47
CALCRL Q16602 13/20 0.46
ADM2 Q7Z4H4 5/20 0.45
RAMP1 O60894 4/20 0.44
CALCB P10092 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17881436 1.00 CALCA (0.47) CALCACALCRLADM2RAMP1CALCB
SCHEMBL13272686 0.86 ADM2 (0.49) CALCRLADM2RAMP1CALCB
SCHEMBL2056346 0.85 CALCA (0.48) CALCACALCRLADM2RAMP1CALCB
SCHEMBL24962033 0.85 CALCA (0.48) CALCACALCRLADM2RAMP1CALCB
SCHEMBL837503 0.85 ADM2 (0.49) CALCACALCRLADM2RAMP1CALCB
SCHEMBL17881601 0.84 ADM2 (0.55) CALCRLADM2CALCB
SCHEMBL260489 0.84 ADM2 (0.55) CALCRLADM2CALCB
SCHEMBL1818060 0.84 ADM2 (0.55) CALCRLADM2CALCB
SCHEMBL22796652 0.82 CALCA (0.48) CALCACALCRLADM2RAMP1CALCB
SCHEMBL22774650 0.82 CALCA (0.48) CALCACALCRLADM2RAMP1CALCB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143266-B2 Aryl heterocyclic CGRP receptor antagonists Merck, Sharp & Dohme Corp (US) 2012-03-27 US disclosed