SCHEMBL8463240

SCHEMBL8463240

CCOC(=O)c1cn(C)c([S+]([O-])CCC=C(F)F)n1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.37
GABRA2 P47869 6/20 0.37
GABRB2 P47870 6/20 0.37
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
CYP1A2 P05177 1/20 0.36
RAB9A P51151 5/20 0.33
NPC1 O15118 4/20 0.33
RXFP1 Q9HBX9 1/20 0.33
PTGS2 P35354 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
MLYCD O95822 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8464878 0.74 GAA (0.38) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL8466902 0.74 GAA (0.38) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL9046316 0.70 KDM4E (0.35) KDM4EALDH1A1POLBHPGDCYP1A2
SCHEMBL16519359 0.68 CYP1A2 (0.53) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL5140534 0.67 MITF (0.49) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL1001660 0.66 CYP1A2 (0.50) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL25658525 0.66 CYP1A2 (0.50) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL16268836 0.66 CYP1A2 (0.50) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL26311965 0.66 GAA (0.52) GAAGABRA2GABRB2KDM4EALDH1A1
SCHEMBL5041765 0.64 CYP1A2 (0.47) GAAGABRA2GABRB2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5912243-A NOVEL COMPOUNDS FOR CONTROLLING NEMATODES, INSECT OR ACARID PESTS ZENECA LIMITED (GB) 1999-06-15 US disclosed
US-5705516-A NEMATOCIDES, INSECTICIDES, ACARICIDES ZENECA LIMITED (GB) 1998-01-06 US disclosed
WO-1995024403-A1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY ZENECA LIMITED (GB) 1995-09-14 WO disclosed