SCHEMBL8464285

SCHEMBL8464285

CNc1ncnc2c1ncn2CCCCCOC(=O)N[C@@H](CCCNC(=N)N)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY1 P47900 2/20 0.43
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
ADCY5 O95622 4/20 0.36
DOT1L Q8TEK3 2/20 0.35
PRMT1 Q99873 1/20 0.35
MARS1 P56192 1/20 0.35
IARS1 P41252 1/20 0.34
HDAC1 Q13547 4/20 0.34
HDAC2 Q92769 4/20 0.34
PDE5A O76074 1/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE1C Q14123 1/20 0.34
PDE3A Q14432 1/20 0.34
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8467074 1.00 P2RY1 (0.43) P2RY1PDE4APDE4BPDE4CPDE4D
SCHEMBL8467662 0.93 ADCY5 (0.36) P2RY1ADCY5MARS1IARS1HDAC1
SCHEMBL8465925 0.93 ADCY5 (0.36) P2RY1ADCY5MARS1IARS1HDAC1
SCHEMBL8466911 0.90 ADCY5 (0.37) P2RY1ADCY5MARS1HDAC1HDAC2
SCHEMBL8466600 0.90 ADCY5 (0.47) ADCY5PDE3A
SCHEMBL8465859 0.90 ADCY5 (0.47) ADCY5PDE3A
SCHEMBL8464093 0.90 DOT1L (0.39) ADCY5DOT1LMARS1IARS1
SCHEMBL8464786 0.90 DOT1L (0.39) ADCY5DOT1LMARS1IARS1
SCHEMBL8467135 0.90 TAAR1 (0.42) P2RY1ADCY5MARS1IARS1
SCHEMBL8466905 0.89 ADCY5 (0.36) ADCY5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994361-A ANTITUMOR, ANTICANCER AGENT BIOCHEM PHARMA (CA) 1999-11-30 US claimed