SCHEMBL8465103

SCHEMBL8465103

Cc1cccc2c1C(=O)c1c(nc3ccccn13)C2=O

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.69
HSP90AB1 P08238 1/20 0.69
DPP4 P27487 1/20 0.51
MAPK13 O15264 2/20 0.46
MAPK12 P53778 2/20 0.46
MAPK11 Q15759 2/20 0.46
MAPK14 Q16539 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8464963 0.95 HSP90AA1 (0.69) HSP90AA1HSP90AB1DPP4MAPK13MAPK12
SCHEMBL8465070 0.89 HSP90AA1 (0.61) HSP90AA1HSP90AB1DPP4MAPK13MAPK12
SCHEMBL8466674 0.89 HSP90AA1 (0.61) HSP90AA1HSP90AB1DPP4MAPK13MAPK12
SCHEMBL8464939 0.84 HSP90AA1 (0.69) HSP90AA1HSP90AB1
SCHEMBL1274825 0.82 HSP90AA1 (1.00) HSP90AA1HSP90AB1
SCHEMBL8466658 0.81 HSP90AA1 (0.44) HSP90AA1HSP90AB1
SCHEMBL8466603 0.80 HSP90AA1 (0.63) HSP90AA1HSP90AB1
SCHEMBL8465262 0.78 HSP90AA1 (0.69) HSP90AA1HSP90AB1
SCHEMBL31237216 0.76 HSP90AA1 (0.61) HSP90AA1HSP90AB1MAPK13MAPK12MAPK11
SCHEMBL8465132 0.76 HSP90AA1 (0.61) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981544-A Mono-- or diketone tetracyclic derivatives and therapeutical uses thereof LABORATOIRE INNOTHERA (FR) 1999-11-09 US claimed
US-5981544-A Mono-- or diketone tetracyclic derivatives and therapeutical uses thereof LABORATOIRE INNOTHERA (FR) 1999-11-09 US disclosed