SCHEMBL8466930

SCHEMBL8466930

CSc1ncnc2c1ncn2CCCCCO

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.72
TSHR P16473 1/20 0.72
ADORA2A P29274 4/20 0.56
ADCY1 Q08828 1/20 0.50
ADORA1 P30542 2/20 0.48
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ADCY5 O95622 3/20 0.43
TK1 P04183 1/20 0.43
CYP2D6 P10635 1/20 0.42
MAPK1 P28482 1/20 0.42
ADORA2B P29275 1/20 0.41
TLR9 Q9NR96 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10362340 0.80 ADORA2A (0.61) CYP1A2TSHRADORA2AADCY1ADORA1
SCHEMBL8464071 0.78 ADORA2A (0.60) CYP1A2TSHRADORA2AADCY1ADORA1
SCHEMBL8467390 0.78 ADORA2A (0.88) ADORA2AADCY1ADORA1ADCY5ADORA2B
SCHEMBL8467138 0.78 ADORA2A (0.60) CYP1A2TSHRADORA2AADCY1ADORA1
SCHEMBL8467559 0.78 ADORA2A (0.60) CYP1A2TSHRADORA2AADCY1ADORA1
SCHEMBL7812370 0.78 ADORA2A (0.63) CYP1A2TSHRADORA2AADCY1ADORA1
SCHEMBL8467638 0.78 ADORA2A (0.56) ADORA2AADCY1ADORA1ADCY5
SCHEMBL8465881 0.78 ADORA2A (0.56) CYP1A2TSHRADORA2AADCY1ADORA1
SCHEMBL8464512 0.78 CYP1A2 (0.73) CYP1A2TSHRADORA2AADCY1ADORA1
SCHEMBL8464772 0.78 CYP1A2 (0.73) CYP1A2TSHRADORA2AADCY1ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994361-A ANTITUMOR, ANTICANCER AGENT BIOCHEM PHARMA (CA) 1999-11-30 US claimed