Colchicine

Colchicine

SCHEMBL8469

COc1cc2c(c(OC)c1OC)-c1ccc(OC)c(=O)cc1[C@@H](NC(C)=O)CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8

The experimentally established mechanism targets of Colchicine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 known ✓ Q9H4B7 7/20 1.00
TUBB4A known ✓ P04350 4/20 1.00
TUBB known ✓ P07437 4/20 1.00
TUBA3C known ✓ P0DPH7 4/20 1.00
TUBA1B known ✓ P68363 4/20 1.00
TUBA4A known ✓ P68366 4/20 1.00
TUBB4B known ✓ P68371 4/20 1.00
TUBB3 known ✓ Q13509 4/20 1.00
TUBB2A known ✓ Q13885 4/20 1.00
TUBB8 known ✓ Q3ZCM7 4/20 1.00
TUBA3E known ✓ Q6PEY2 4/20 1.00
TUBA1A known ✓ Q71U36 4/20 1.00
TUBA1C known ✓ Q9BQE3 4/20 1.00
TUBB6 known ✓ Q9BUF5 4/20 1.00
TUBB2B known ✓ Q9BVA1 4/20 1.00
LMNA P02545 3/20 1.00
CYP2C9 P11712 3/20 1.00
TSHR P16473 2/20 1.00
KMT2A Q03164 2/20 1.00
MITF O75030 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Colchicine SCHEMBL29374654 1.00 TUBB1 (1.00) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL1658120 1.00 TUBB1 (1.00) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL29376116 1.00 TUBB1 (1.00) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL15521905 1.00 TUBB1 (1.00) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL8669234 1.00 TUBB1 (1.00) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL675246 1.00 TUBB1 (1.00) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL2006815 0.99 TUBB1 (0.98) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL7617204 0.99 TUBB1 (0.98) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL2005815 0.99 TUBB1 (0.98) TUBB1TUBB4ATUBBTUBA3CTUBA1B
Colchicine SCHEMBL28039025 0.99 TUBB1 (0.98) TUBB1TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 103315 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144890-A1 ANTIBODY DRUG CONJUGATE COMPRISING NMT INHIBITOR CONJUGATED TO AN ANTIBODY MyricX Pharma Limited (GB) 2026-05-28 US claimed
EP-4228644-B1 N-[4-[1-(1,4-DIOXASPIRO[4.5]DEC-8-YL)-4-(8-OXA-3-AZABICYCLO[3.2.1]OCT-3-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-6-YL]PHENYL]-N'-METHYLUREA FOR USE IN THE TREATMENT OF COVID19 NANTCELL INC (US) 2026-05-27 EP claimed
CN-120738280-B Haploid induction line-based plant genetic transformation method INSTITUTE OF CROP SCIENCES, CHINESE ACADEMY OF AGRICULTURAL SCIENCES (CN) 2026-05-26 CN claimed
CN-120208981-B Colchicine binding site inhibitor prodrug, nano-drug and preparation and application thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2026-05-26 CN claimed
CN-122075699-A Application of calcium activated chloride channel AN01/TMEM16A in preventing and treating atherosclerosis 2026-05-26 CN claimed
CN-122080895-A Polyglycolic acid composition and preparation method thereof, biodegradable polyester material and application thereof, and PGA temporary plugging ball and preparation method thereof 2026-05-26 CN claimed
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
US-20260137686-A1 SOLID PHARMACEUTICAL FORMULATION OF PARP INHIBITORS AND USE THEREOF IMPACT THERAPEUTICS SHANGHAI INC (CN) 2026-05-21 US claimed
US-20260137041-A1 SIMULTANEOUS GENE EDITING AND HAPLOID INDUCTION SYNGENTA CROP PROTECTION AG (CH) 2026-05-21 US claimed
US-20260138973-A1 SUBSTITUTED PYRIDINES FOR USE IN TREATING OR PREVENTING INFLAMMATORY DISEASES OR DISEASES ASSOCIATED WITH AN UNDESIRABLE IMMUNE RESPONSE SITRYX THERAPEUTICS LTD (GB) 2026-05-21 US claimed
US-4309415-A LINOLENIC ACID OR DERIVATIVE WITH MATERIAL WHICH ENHANCES BIOSYNTHESIS OF THROMBOXANE A2 VERRONMAY LIMITED (GB) 1982-01-05 US claimed
EP-0037175-A1 Pharmaceutical compositions EFAMOL LIMITED (GB) 1981-10-07 EP claimed
EP-0035856-A2 Pharmaceutical and dietary compositions EFAMOL LIMITED (GB) 1981-09-16 EP claimed
EP-0019423-A1 Pharmaceutical and dietary composition comprising gamma-linolenic acids EFAMOL LIMITED (GB) 1980-11-26 EP claimed
US-4190673-A Colchicine ophthalmic composition and method of use NELSON RESEARCH & DEVELOPMENT COMPANY (US) 1980-02-26 US claimed
EP-0004770-A2 Pharmaceutical and dietary composition comprising gamma-linolenic acids EFAMOL LIMITED (GB) 1979-10-17 EP claimed
US-4147767-A CROSSLINKED WITH FORMALDEHYDE OR GLUTARALDEHYDE MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1979-04-03 US claimed
US-4102079-A Method of breeding new varieties of the first filial generation plant KATAOKA SETSUO 1978-07-25 US claimed
US-4014334-A Laminated osmotic system for dispensing beneficial agent ALZA CORPORATION (US) 1977-03-29 US claimed
US-4008719-A Osmotic system having laminar arrangement for programming delivery of active agent ALZA CORPORATION (US) 1977-02-22 US claimed