SCHEMBL8470256

SCHEMBL8470256

Cc1nn(C)c(C)c1-n1ccnc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.37
HSD17B10 Q99714 2/20 0.35
NFKB1 P19838 1/20 0.35
QPCT Q16769 1/20 0.35
QPCTL Q9NXS2 1/20 0.35
CYP19A1 P11511 1/20 0.35
MAPT P10636 4/20 0.35
LMNA P02545 4/20 0.35
ENPP2 Q13822 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
NOTUM Q6P988 1/20 0.35
CYP2A6 P11509 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
CYP1A2 P05177 3/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
ALDH1A1 P00352 2/20 0.33
MITF O75030 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16923117 0.72 CYP3A4 (0.54) CYP3A4HSD17B10NFKB1QPCTQPCTL
SCHEMBL13683147 0.71 NOTUM (0.41) CYP3A4HSD17B10NFKB1QPCTQPCTL
SCHEMBL1231062 0.67 CYP11B1 (0.50) CYP3A4HSD17B10CYP19A1MAPTLMNA
SCHEMBL7649005 0.67 CYP3A4 (0.50) CYP3A4HSD17B10CYP19A1MAPTLMNA
SCHEMBL22366437 0.67 CYP3A4 (0.51) CYP3A4CYP19A1MAPTLMNAENPP2
Bromide SCHEMBL28821466 0.65 CYP11B1 (0.49) CYP3A4HSD17B10MAPTLMNAENPP2
Bromide SCHEMBL12481601 0.65 CYP11B1 (0.49) CYP3A4HSD17B10MAPTLMNAENPP2
Silver SCHEMBL28021712 0.65 CYP11B1 (0.49) CYP3A4HSD17B10MAPTLMNAENPP2
Hydrochloric Acid SCHEMBL28521741 0.65 CYP3A4 (0.48) CYP3A4HSD17B10CYP19A1MAPTLMNA
Hydrochloric Acid SCHEMBL5168891 0.65 CYP11B1 (0.49) CYP3A4HSD17B10MAPTLMNAENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO claimed