SCHEMBL8470768

SCHEMBL8470768

O=C(O)CSCc1cccc(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.60
ALDH1A1 P00352 4/20 0.58
TDP1 Q9NUW8 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
HPGD P15428 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
KMT2A Q03164 1/20 0.53
IDO1 P14902 2/20 0.50
KDM4E B2RXH2 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
PTPRC P08575 1/20 0.50
PTPRG P23470 1/20 0.50
THRB P10828 1/20 0.49
MAPT P10636 1/20 0.49
CTBP2 P56545 1/20 0.49
TP53 P04637 1/20 0.48
HCAR2 Q8TDS4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31366769 0.81 IDO1 (0.58) ALDH1A1HPGDSMN1; SMN2IDO1CYP3A4
SCHEMBL3905722 0.81 CYP1A2 (0.62) CYP1A2SMN1; SMN2IDO1KDM4ECYP2C19
SCHEMBL1635769 0.79 CYP1A2 (0.60) CYP1A2ALDH1A1TDP1L3MBTL1SMN1; SMN2
SCHEMBL15083077 0.79 CYP1A2 (0.65) CYP1A2ALDH1A1KDM4ECYP3A4CYP2D6
SCHEMBL2208069 0.79 CYP1A2 (0.60) CYP1A2ALDH1A1SMN1; SMN2KMT2AIDO1
SCHEMBL3910561 0.79 CYP1A2 (0.60) CYP1A2ALDH1A1KDM4ECYP3A4CYP2D6
SCHEMBL30050703 0.79 CYP1A2 (0.60) CYP1A2ALDH1A1KDM4ECYP3A4CYP2D6
SCHEMBL10419640 0.79 CYP1A2 (0.65) CYP1A2ALDH1A1L3MBTL1HPGDKMT2A
SCHEMBL499117 0.79 CYP2C19 (0.64) CYP1A2ALDH1A1SMN1; SMN2CYP2C19MAPT
Hydrochloric Acid SCHEMBL3909181 0.78 CYP1A2 (0.59) CYP1A2ALDH1A1KMT2AKDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110229333-A A kind of synthetic method of new type polyimide 湘潭大学 2019-09-13 CN disclosed
US-5886016-A ANTIINFLAMMATORY AGENT WITH MINIMAL SIDE EFFECTS FOR TREATING ARTHRITIS G.D. SEARLE & CO. (US) 1999-03-23 US disclosed
US-5670532-A Pyrazolyl derivatives for the treatment of inflammation G. D. SEARLE & CO. (US) 1997-09-23 US disclosed
US-5565482-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS G.D. SEARLE & CO. (US) 1996-10-15 US disclosed
US-5547975-A ANTIARTHRIC AGENTS, ANALGESICS AND ANTIPYRETICS; INHIBITORS OF CYCLOOXYGENASE II; SIDE EFFECT REDUCTION G.D. SEARLE & CO. 1996-08-20 US disclosed
WO-1996009304-A1 BENZOPYRANOPYRAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed