SCHEMBL8470920

SCHEMBL8470920

CN(CCCF)C(=O)c1cc2ccccc2c(-c2ccccc2I)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSPO P30536 7/20 0.64
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
NR1I3 Q14994 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8474804 0.94 TSPO (0.65) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8474388 0.90 TSPO (0.65) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8470616 0.86 TSPO (0.60) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8473026 0.85 TSPO (0.46) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8474046 0.84 TSPO (0.47) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8523967 0.83 TSPO (0.61) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8470697 0.83 TSPO (0.44) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8470604 0.82 TSPO (0.56) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8473060 0.82 TSPO (0.79) TSPOMEN1KMT2ACYP3A4CYP2C9
SCHEMBL8474523 0.81 TSPO (0.45) TSPOMEN1KMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998624-A MEDICAL DIAGNOSIS; BINDING TO SITE OF INJURY, INFLAMMATION EMORY UNIVERSITY (US) 1999-12-07 US disclosed
WO-1998049900-A1 HALOISOQUINOLINE CARBOXAMIDE EMORY UNIVERSITY (US) 1998-11-12 WO disclosed