SCHEMBL8471964

SCHEMBL8471964

COc1ccc(-c2ccccc2)c(NC(=O)C(C)(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
KDM4E B2RXH2 6/20 0.52
L3MBTL1 Q9Y468 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
KMT2A Q03164 2/20 0.52
GAA P10253 4/20 0.51
MAPT P10636 3/20 0.51
CHRM3 P20309 1/20 0.49
TACR1 P25103 1/20 0.49
LMNA P02545 3/20 0.47
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TOP2A P11388 1/20 0.46
POLB P06746 1/20 0.46
ADORA1 P30542 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
HDAC8 Q9BY41 1/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5106389 0.85 KDM4E (0.53) ALDH1A1KDM4EL3MBTL1NPSR1KMT2A
SCHEMBL17206259 0.84 KDM4E (0.52) ALDH1A1KDM4EL3MBTL1NPSR1KMT2A
SCHEMBL8473546 0.84 CHRM3 (0.46) ALDH1A1KDM4EL3MBTL1NPSR1KMT2A
SCHEMBL14447514 0.80 TACR1 (0.64) ALDH1A1KDM4EKMT2AMAPTTACR1
SCHEMBL1663014 0.78 AKR1C3 (0.60) KDM4ENPSR1KMT2AMEN1
SCHEMBL4013508 0.78 GAA (0.56) KDM4ENPSR1KMT2AGAAMAPT
SCHEMBL5226002 0.77 TDP1 (0.54) KDM4ENPSR1KMT2AGAAMAPT
SCHEMBL18415466 0.77 ALDH1A1 (0.53) ALDH1A1KDM4EL3MBTL1NPSR1KMT2A
SCHEMBL16438566 0.77 ALDH1A1 (0.53) ALDH1A1KDM4EL3MBTL1NPSR1KMT2A
SCHEMBL30076369 0.77 ALDH1A1 (0.47) ALDH1A1KDM4ENPSR1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948817-A Polycyclic ethyl alkylamide melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1999-09-07 US disclosed
WO-1998038991-A1 POLYCYCLIC ETHYL ALKYLAMIDE MELATONERGIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-09-11 WO disclosed