SCHEMBL8471981

SCHEMBL8471981

COc1ccc(N2CCN(CCO)C2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.56
DRD2 P14416 8/20 0.51
DRD3 P35462 8/20 0.51
CYP1A1 P04798 5/20 0.51
PKM P14618 1/20 0.49
DPP4 P27487 1/20 0.48
KCNH2 Q12809 3/20 0.47
S1PR1 P21453 1/20 0.43
NOX4 Q9NPH5 1/20 0.43
RAB9A P51151 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6220245 0.85 HDAC1 (0.56) HDAC1DRD2DRD3CYP1A1PKM
SCHEMBL14734293 0.83 HDAC1 (0.56) HDAC1DRD2DRD3CYP1A1PKM
SCHEMBL27968105 0.82 HTR2C (0.55) DRD2DRD3CYP1A1DPP4KCNH2
SCHEMBL3714292 0.82 DRD2 (0.61) HDAC1DRD2DRD3CYP1A1PKM
SCHEMBL2199747 0.81 HDAC1 (0.49) HDAC1DRD2DRD3CYP1A1PKM
SCHEMBL17080505 0.80 DRD2 (0.48) HDAC1DRD2DRD3CYP1A1KCNH2
SCHEMBL17080578 0.80 DRD2 (0.48) HDAC1DRD2DRD3CYP1A1KCNH2
SCHEMBL10498393 0.80 CYP1A1 (0.64) HDAC1DRD2DRD3CYP1A1S1PR1
SCHEMBL5659037 0.80 DRD2 (0.65) HDAC1DRD2DRD3KCNH2RAB9A
SCHEMBL27734214 0.79 HDAC1 (0.53) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990139-A 2,5-DIOXO-4-(PYRIDYL OR PHENYL-(N-HETEROCYCLE(C4N,C3N2))-ALKYLENOXY-(1,4-PHENYLENE) -)THIADIAZOLIDINES; ANTIDIABETIC AND -LIPEMIC AGENTS; SIDE EFFECT REDUCTION TAIHO PHARMACEUTICAL CO., LTD. (JP) 1999-11-23 US disclosed