SCHEMBL8477000

SCHEMBL8477000

COc1ccc(CC2C3=C(CCCC3)CCN2C=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
PDE4D Q08499 2/20 0.39
MTNR1B P49286 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.36
MTNR1A P48039 1/20 0.35
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11360939 0.85 CTSK (0.38) MTNR1BHRH3MMP9MTNR1A
SCHEMBL11366916 0.83 CAPN1 (0.43) ALDH1A1
SCHEMBL2067120 0.82 BCHE (0.53) CYP2D6BCHEACHEALDH1A1HRH3
SCHEMBL16596978 0.82 BCHE (0.53) CYP2D6BCHEACHEALDH1A1HRH3
SCHEMBL6545035 0.79 CYP3A4 (0.48) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL9151971 0.78 CYP2D6 (0.61) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL8951697 0.78 CYP3A4 (0.38) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL11757293 0.78 CYP2D6 (0.61) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL11447599 0.76 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C19BCHEACHE
SCHEMBL16596996 0.76 BCHE (0.32) CYP3A4CYP2D6CYP2C19BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5905153-A INTERMEDIATES FOR MANUFACTURE OF DEXTROMETHORPHAN ROCHE VITAMINS INC. (US) 1999-05-18 US disclosed
US-4052389-A DERIVATIVES OF 9,10-DIHYDROXY-1-(P-ALKOXYBENZYL)-PERHYDROISOQUINOLINE OXAZINE-3-ONE BRISTOL-MYERS COMPANY (US) 1977-10-04 US disclosed