SCHEMBL8477200

SCHEMBL8477200

OC(CCc1cccnc1)CSc1cccc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPK1 P28482 1/20 0.39
HTR2C P28335 1/20 0.39
POLB P06746 1/20 0.38
CYP3A4 P08684 3/20 0.38
CHRNA7 P36544 2/20 0.38
HPGD P15428 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PSMD14 O00487 1/20 0.36
STAMBP O95630 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483322 0.89 ALDH1A1 (0.40) ALDH1A1LMNAKDM4EMAPK1HTR2C
SCHEMBL6947292 0.79 HTT (0.46) ALDH1A1KDM4ECYP3A4CHRNA7CYP1A2
SCHEMBL8479651 0.79 BACE1 (0.50) ALDH1A1LMNACYP3A4CYP2D6CYP2C9
SCHEMBL8550527 0.77 BACE1 (0.48) ALDH1A1LMNACYP3A4CYP2D6CYP2C9
SCHEMBL8551871 0.77 NAMPT (0.39) ALDH1A1LMNAKDM4EMAPK1POLB
SCHEMBL23391645 0.77 BACE1 (0.45) ALDH1A1LMNAKDM4EMAPK1CYP1A2
SCHEMBL29715998 0.77 BACE1 (0.45) ALDH1A1LMNAKDM4EMAPK1CYP1A2
SCHEMBL8549887 0.75 BACE1 (0.41) MAPK1HTR2CPOLBCYP3A4CYP1A2
SCHEMBL8482634 0.75 BACE1 (0.48) KDM4ECHRNA7SMN1; SMN2
SCHEMBL8479405 0.75 NPC1 (0.44) LMNAKDM4EPOLBCHRNA7SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977105-A Compounds ASTRA PHARMAEUTICALS LTD. (GB) 1999-11-02 US disclosed
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed