SCHEMBL8477408

SCHEMBL8477408

OC(Cc1cc[c]cc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.51
CYP2C19 P33261 3/20 0.51
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 1/20 0.51
HIF1A Q16665 1/20 0.51
KCNA5 P22460 1/20 0.51
CYP2D6 P10635 2/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
FDPS P14324 1/20 0.37
CHRM2 P08172 4/20 0.36
CHRM4 P08173 4/20 0.36
CHRM5 P08912 4/20 0.36
CHRM1 P11229 4/20 0.36
CHRM3 P20309 4/20 0.36
LMNA P02545 1/20 0.36
HTR1A P08908 1/20 0.36
OPRM1 P35372 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27969023 0.85 CYP1A2 (0.45) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
SCHEMBL912792 0.85 CYP2C9 (0.67) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
Phosphine SCHEMBL11171774 0.83 CYP2C9 (0.64) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
SCHEMBL8474675 0.81 EBP (0.43) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
SCHEMBL9069470 0.79 CYP2C9 (0.60) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
SCHEMBL8480984 0.77 LMNA (0.44) MEN1KMT2ASMN1; SMN2LMNAKCNH2
SCHEMBL5873436 0.76 HTT (0.53) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
SCHEMBL8974025 0.76 ESR1 (0.47) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
SCHEMBL5347146 0.76 CYP2C9 (0.56) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A
SCHEMBL8480296 0.76 TAAR1 (0.42) CYP2C9CYP2C19CYP1A2CYP3A4HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6004988-A Carboxylic acid derivatives, their preparation and their use BASF AKTIENGESELLSCHAFT (DE) 1999-12-21 US disclosed
US-4855290-A Derivatives of quinuclidine STATE OF ISRAEL, REPRESENTED BY PRIME MINISTER'S OFFICE, ISRAEL INSTITUTE FOR BIOLOGICAL RESEARCH (IL) 1989-08-08 US disclosed