SCHEMBL8477589

SCHEMBL8477589

C[C@@H](C(O)CCC(=O)OC(C)(C)C)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.41
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
KLK5 Q9Y337 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CTSL P07711 2/20 0.38
CTSB P07858 2/20 0.38
CTSS P25774 2/20 0.38
PSEN1 P49768 2/20 0.38
PSEN2 P49810 2/20 0.38
APH1B Q8WW43 2/20 0.38
NCSTN Q92542 2/20 0.38
APH1A Q96BI3 2/20 0.38
PSENEN Q9NZ42 2/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8475218 1.00 AKT1 (0.41) AKT1JAK2JAK1KLK5MEN1
SCHEMBL29283791 0.81 AKT1 (0.42) AKT1JAK2JAK1MEN1KMT2A
SCHEMBL2863308 0.80 AKT1 (0.41) AKT1MEN1KMT2AHTTL3MBTL1
SCHEMBL29283793 0.80 AKT1 (0.41) AKT1KLK5MEN1KMT2AHTT
SCHEMBL8476974 0.79 AKT1 (0.43) AKT1MEN1KMT2AHTTL3MBTL1
SCHEMBL13109078 0.76 AKT1 (0.37) AKT1JAK2JAK1MEN1KMT2A
SCHEMBL15153449 0.75 MAPT (0.39) MEN1KMT2ACTSLCTSS
SCHEMBL14728040 0.75 MAPT (0.39) MEN1KMT2ACTSLCTSS
SCHEMBL15153451 0.75 MAPT (0.39) MEN1KMT2ACTSLCTSS
SCHEMBL10453045 0.74 ABCB1 (0.50) MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990341-A Diastereoselective synthesis hydroxyethylene dipeptide isosteres EMORY UNIVERSITY (US) 1999-11-23 US disclosed
US-5587514-A Diastereoselective synthesis of hydroxyethylene dipeptide isosteres EMORY UNIVERSITY (US) 1996-12-24 US disclosed