SCHEMBL8478753

SCHEMBL8478753

C/C(=C/C(=O)O)c1cnccn1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
NAPRT Q6XQN6 1/20 0.57
HCAR2 Q8TDS4 1/20 0.57
ADORA3 P0DMS8 1/20 0.50
TSHR P16473 1/20 0.50
MC4R P32245 1/20 0.50
ADRA1A P35348 1/20 0.50
MC3R P41968 1/20 0.50
NPC1 O15118 6/20 0.46
RAB9A P51151 6/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
MAPT P10636 1/20 0.46
GAA P10253 2/20 0.45
TBXAS1 P24557 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8478756 1.00 KDM4E (0.57) KDM4ENAPRTHCAR2ADORA3TSHR
SCHEMBL8779941 0.81 KDM4E (0.47) KDM4ENAPRTHCAR2ADORA3TSHR
SCHEMBL8779937 0.81 KDM4E (0.47) KDM4ENAPRTHCAR2ADORA3TSHR
SCHEMBL7702024 0.78 KDM4E (0.50) KDM4ENAPRTHCAR2ADORA3TSHR
SCHEMBL27313644 0.78 KDM4E (0.57) KDM4ENAPRTHCAR2ADORA3TSHR
SCHEMBL29993937 0.76
SCHEMBL78340 0.76
SCHEMBL29742199 0.74 KDM4E (0.61) KDM4ENAPRTHCAR2ADORA3TSHR
Pyrazine SCHEMBL15798805 0.74 KDM4E (0.61) KDM4ENAPRTHCAR2ADORA3TSHR
Pyrazinoic Acid SCHEMBL29651929 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939268-A DIELS-ALDER REACTION PRODUCT OF A DIENE AND A DIENOPHILE; CHEMICAL INTERMEDIATES FOR DRUGS, SOLID PHASE SYNTHESIS THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US claimed
US-5939268-A DIELS-ALDER REACTION PRODUCT OF A DIENE AND A DIENOPHILE; CHEMICAL INTERMEDIATES FOR DRUGS, SOLID PHASE SYNTHESIS THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US disclosed
EP-0773953-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS INSTITUTE (US) 1997-05-21 EP disclosed
WO-1996003424-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS RESEARCH INSTITUTE (US) 1996-02-08 WO disclosed