SCHEMBL27313644

SCHEMBL27313644

O=C(O)/C=C(/C(=O)O)c1cnccn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.57
NAPRT Q6XQN6 1/20 0.57
HCAR2 Q8TDS4 1/20 0.57
TSHR P16473 2/20 0.50
ADORA3 P0DMS8 1/20 0.50
MC4R P32245 1/20 0.50
ADRA1A P35348 1/20 0.50
MC3R P41968 1/20 0.50
BAZ2B Q9UIF8 1/20 0.41
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KMT2A Q03164 3/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8478753 0.78 KDM4E (0.57) KDM4ENAPRTHCAR2TSHRADORA3
SCHEMBL8478756 0.78 KDM4E (0.57) KDM4ENAPRTHCAR2TSHRADORA3
SCHEMBL7091828 0.76 KMT2A (0.56) KDM4ENAPRTHCAR2TSHRADORA3
SCHEMBL27330261 0.74 LMNA (0.57) KDM4ENAPRTNPC1RAB9ASMN1; SMN2
SCHEMBL11538095 0.74 LMNA (0.57) KDM4ENAPRTNPC1RAB9ASMN1; SMN2
SCHEMBL27497486 0.74 KDM4E (0.68) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL23757 0.73
Pyrazinoic Acid SCHEMBL29651929 0.73
SCHEMBL19614365 0.73 GRM5 (0.41) HCAR2
SCHEMBL23230628 0.71 KDM4E (0.53) KDM4ENAPRTHCAR2TSHRADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1030986-C Pyrrolopyrazine HOFFMANN LA ROCHE (CH) 1996-02-14 CN disclosed
CN-1068328-A PYRROLOPYRAZINE HOFFMANN LA ROCHE (CH) 1993-01-27 CN disclosed