SCHEMBL8479166

SCHEMBL8479166

Clc1cc2[nH][c]cc2cc1Br

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.52
AHR P35869 2/20 0.37
HAVCR2 Q8TDQ0 1/20 0.31
AXL P30530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2715277 0.81 ALDH1A1 (0.39) CSNK2A1
SCHEMBL22462465 0.81 ALDH1A1 (0.31) CSNK2A1
SCHEMBL10179972 0.68 CSNK2A1 (1.00) CSNK2A1AHR
SCHEMBL22655868 0.67 AXL (0.56) CSNK2A1AXL
SCHEMBL14889487 0.67 CSNK2A1 (0.48) CSNK2A1AHRHAVCR2
SCHEMBL17351236 0.67 CSNK2A1 (0.48) CSNK2A1AHRHAVCR2AXL
SCHEMBL3850787 0.66 AHR (0.58) CSNK2A1AHR
SCHEMBL207489 0.64 F7 (0.50) AHRHAVCR2
SCHEMBL207737 0.64 CYP2A6 (0.50) CSNK2A1AHR
SCHEMBL11282194 0.64 AHR (0.55) CSNK2A1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925647-A TREATMENT OF INSULIN NON-INSULIN DEPENDENT DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1999-07-20 US disclosed
US-5681958-A TREATMENT OF DIABETES SHAMAN PHARMACEUTICALS, INC. (US) 1997-10-28 US disclosed
WO-1996010015-A1 CRYPTOLEPINE ANALOGS WITH HYPOGLYCEMIC ACTIVITY SHAMAN PHARMACEUTICALS, INC. (US) 1996-04-04 WO disclosed