SCHEMBL8480429

SCHEMBL8480429

Nc1c(-c2cc(Cl)ccc2O)c2ccc(C(F)(F)F)cc2[nH]c1=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 10/20 0.62
CYP3A4 P08684 4/20 0.62
CYP2C19 P33261 4/20 0.62
CYP2D6 P10635 2/20 0.62
CYP1A2 P05177 1/20 0.62
BIRC5 O15392 1/20 0.46
JUN P05412 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
PIM1 P11309 2/20 0.46
CDK2 P24941 2/20 0.46
CLK2 P49760 2/20 0.46
GSK3B P49841 2/20 0.46
CAMK2B Q13554 2/20 0.46
CAMK2G Q13555 2/20 0.46
CAMK2D Q13557 2/20 0.46
DYRK1A Q13627 2/20 0.46
CDC42BPA Q5VT25 2/20 0.46
PLK3 Q9H4B4 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8479190 0.92 CYP2C9 (0.73) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6545364 0.88 CYP2C9 (0.62) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
Formic Acid SCHEMBL8479075 0.88 CYP2C9 (0.68) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL3275049 0.85 CYP2C9 (0.86) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL8476895 0.84 CYP2C9 (0.63) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL8476391 0.83 CYP2C9 (0.53) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL27637829 0.82 CYP2C9 (0.57) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL8475930 0.81 GSK3B (0.54) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL8479083 0.81 GSK3B (0.56) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL7485392 0.80 PIM1 (0.63) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972961-A ANTIISCHEMIC AGENTS; ANTICONVULSANTS; HEADACHES; SEXUAL DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-10-26 US disclosed