SCHEMBL8483753

SCHEMBL8483753

CN(C)CCn1nc2c3c(c([N+](=O)[O-])ccc31)Sc1cnccc1-2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.44
TOP2A P11388 4/20 0.35
TOP2B Q02880 2/20 0.35
EGFR P00533 2/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
PABPC1 P11940 1/20 0.33
CCR6 P51684 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487417 0.90 TOP2A (0.44) NQO1TOP2ATOP2BPOLBKMT2A
SCHEMBL10927511 0.87 NQO1 (0.46) NQO1TOP2ATOP2BEGFRMEN1
SCHEMBL8489718 0.87 NQO1 (0.35) NQO1POLBMAPTHTT
SCHEMBL8487874 0.86 NQO1 (0.35) NQO1TOP2ATOP2BMAPTHTT
SCHEMBL8485118 0.83 CYP2D6 (0.36) NQO1TOP2ATOP2BCYP1A2CYP3A4
SCHEMBL8483564 0.82 TOP2A (0.41) NQO1TOP2ATOP2B
SCHEMBL10812237 0.81 NQO1 (0.53) NQO1TOP2ATOP2BEGFRMEN1
SCHEMBL8485482 0.81 NQO1 (0.41) NQO1TOP2ATOP2BEGFRMEN1
SCHEMBL8483509 0.79 NQO1 (0.35) NQO1TOP2ATOP2BMEN1POLB
SCHEMBL8489284 0.78 NQO1 (0.35) NQO1TOP2ATOP2BMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935969-A Pyrido-thiopyrandoinazoles with antitumor activity UNIVERSITY OF VERMONT (US) 1999-08-10 US disclosed